Nonnucleoside reverse transcriptase inhibitors MOA

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Nonnucleoside reverse transcriptase inhibitors MOA

Noncompetitively inhibit reverse transcriptase. Do not require phosphorylation. Toxicity: Rash and hepatotoxicity. CNS sx with efavirenzEfavirenz (CI in pregnancy)NevirapineDelavirdine (CI in pregnancy)